TUG-469

Agonist of FFAR1

Structure

Information

  • FFAR1
  • Agonist
  • up to 1 uM

In Vitro Validations

No in Vitro Validations

In Cell Validations

In Vivo Data

Off-Target Selectivity Assesments

Probe Selectivity in Cell:

No significant activity on the related receptors FFA2 (GPR43) or FFA3 (GPR41). No significant agonist activity at 1 μM on PPARγ

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SERP ratings and comments


SERP Ratings

In Cell Rating
In Model Organisms

(last updated: 26 Feb 2021 )

SERP Ratings

In Cell Rating
In Model Organisms

(last updated: 14 Apr 2021 )