PFI-1

Reagent Authentication Certificate: 
PDF icon Chemical Probes Portal PFI-1.pdf
Protein target name: 
BRD2, BRD3, BRD4, BRDT
Mechanism of action: 
Antagonist

Target Details

Target class: 
Epigenetics
Subclass: 
Bromodomain
Target alias: 
D6S113E, FSH, FSRG1, NAT, O27.1.1, RING3, RNF3, ORFX, RING3L, CAP, HUNK1, HUNKI, MCAP, BRD6, CT9

Probe Details

Chemical Probes Portal ID: 
CPP37
Probe alias: 
QCR-192
SMILES string: 
CN1CC2=C(C=CC(=C2)NS(=O)(=O)C3=CC=CC=C3OC)NC1=O
InChi Key: 
TXZPMHLMPKIUGK-UHFFFAOYSA-N
PAINs evaluation: 
PAINs free

Physico-chemical properties

Solubility - preferred solvent: 
DMSO
Solubility - concentration: 
10 mM
Storage Recommendations
Storage (dry powder): 
2 years -20 oC
Storage sensitivities: 
Avoid freeze-thaw

Primary Reference

External Resources